| Ph.D. | Eric Oblinger, 1997, Catalytica | 
| Helene Fain, 1998, Glaxo Smith-Kline | |
| Jeongbeob Seo, 1999, Array Biopharma | |
| Richard Fornicola, 2001, Albany Molecular | |
| Mario Lozanov, 2001, Albany Molecular | |
| Kande Amarasinghe, 2002, P & G | |
| Maxim Chevliakov, 2002, Cayman Chemicals | |
| Gireesh Mahandru, 2004, Postdoc (University of Indiana, Williams), Phizer | |
| Yike Ni, 2004, Postdoc (Caltech, MacMillan), Wyeth Pharmaceuticals | |
| Andy Skauge, 2004, Postdoc (Texas A & M, Romo) | |
| Minsoo Song, 2004, Postdoc (Temple University, Davis) | |
| Ahmad Al-Dheiby, 2006, Saudi Arabia | |
| Lei Liu, 2006, Shanghai ChemPartner Co. | |
| Christa Chrovian, 2007, Johnson & Johnson | |
| Kanicha sa-ei, 2007, Institute of Chemical and Engineering Sciences, Singapore | |
| Ananda Herath, Postdoc (Burnham Medical Institute) | |
| Mani Chaulagain, Postdoc (Indiana University, Aron) | |
| Refaie Kassab, Postdoc (Virginia Commonwealth University) | |
| Ryan Baxter, 2010, Postdoc (Scripps Research Institute, Blackmond) | |
| Hasnain Malik, 2010, Novartis, Cambridge MA | |
| Grant Sormunen, 2010, Promiliad Biopharma Inc. | |
| Zachary Buchan, 2011, Dow AgroSciences | |
| Wei Li, 2011, Assistant Professor at the University of Toledo | |
| Ben Thompson, 2012, Eastman Chemical Company | |
| Abdur-Rafay Shareef, 2012, Food and Drug Administration | |
| Allison Knauff, 2012, Gonzaga University Visiting Lecturer | |
| Aireal Jenkins, 2012, Postdoc (University of Chicago, Yu) | |
| Solymar Negretti, 2013, Enanta Pharmaceuticals | |
| Taylor Haynes, 2014, Assistant Professor at Caly Poly San Luis Obispo | |
| Jordan Walk, 2014, Lecturer of Chemistry (The College of William and Mary) | |
| Zachary Miller, 2015, Postdoc (University of Wisconsin, Yoon) | |
| Evan Jackson, 2015, Thermo Fisher Scientific | |
| Postdoctoral | Harry Brielmann, 1997, Neurogen | 
| Xiao-Qing Tang, 2000, Mitokor | |
| Erik Kuester, 2001, Memory Pharmaceuticals | |
| Victor Manuel Gutierrez Garcia, 2001-2003, Polaquimia SA de CV | |
| Kandasamy Subburaj, 2001-2003, Arqule | |
| Sanjoy Chowdhury, 2003-2004, Chembiotek | |
| Kirk W. Hering, 2005-2006, Cayman Chemical | |
| Beth Knapp-Reed, 2005-2006, Glaxo Smith-Kline | |
| Scott J. Bader, 2005-2006, Pfizer | |
| John Phillips, 2008-2010, Materia | |
| Katie Partridge, 2010-2012, Eli Lilly | |
| Chris Taylor, 2011-2012 | |
| M.S. Graduate Students | Alexey Savchenko, 1996, Boston Consulting Group | 
| Jean Baptiste Blanc, 1998, Glaxo Smith-Kline | |
| Revathy Venkatachalam, 1998, Astrazeneca | |
| Xin Qi, 2000 | |
| Chongjie Zhu, 2001, Glaxo Smith-Kline | |
| Nicolas Patrin, 2003 | |
| Madduri Srinivasa Rao, 2003, Graduate Student-Purdue University | |
| Gang Liu, 2004, Novartis | |
| Kapil Karki, 2008, Pfizer | |
| Select Undergraduates | Annette Vitale, 1998, Dow Agro (Ph.D. Notre Dame) | 
| Sara Klamo, 1999, Dow Chemical (Ph.D. Caltech) | |
| Keri Muccioli, 1999, Pfizer Global Research | |
| Natalie Giampietro, 2005, Graduate Student - University of Michigan | |
| Thomas Barton, 2007, Graduate Student - University of Texas, Austin | |
| Nicole Harzdorf, 2007, M.S. University of Texas, Austin | |
| Jeannie Kochkodan, 2015, Medical Student, University of Michigan, Ann Arbor |